PD-168077 maleate is a selective dopamine D4 receptor agonist with a Ki of 9 nM. It is for research use only. It shows high selectivity over other D2-like receptor family members and D1-like counterparts, as well as α1, α2, 5-HT1A, and 5-HT2A receptors. It evidences intrinsic activity at the D4 receptor and can induce locomotion in a dose-dependent manner. This product may be used in research related to neurological diseases, neurodegenerative diseases, depression, and Parkinson's disease.
- Selective dopamine D4 receptor agonist
- High selectivity over other receptor types
- Evidences intrinsic activity at the D4 receptor
- Induces locomotion in PD-168077-treated cells
- May be used in research for neurological diseases